Menin-MLL inhibitor 20
CAS No. 2448173-47-3
Menin-MLL inhibitor 20( —— )
Catalog No. M28660 CAS No. 2448173-47-3
Menin-MLL inhibitor 20 is an irreversible menin-MLL interaction inhibitor with antitumor activities (WO2020142557A1, compound 6).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 87 | In Stock |
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| 5MG | 79 | In Stock |
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| 10MG | 130 | In Stock |
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| 25MG | 264 | In Stock |
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| 50MG | 382 | In Stock |
|
| 100MG | 544 | In Stock |
|
| 200MG | 737 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMenin-MLL inhibitor 20
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NoteResearch use only, not for human use.
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Brief DescriptionMenin-MLL inhibitor 20 is an irreversible menin-MLL interaction inhibitor with antitumor activities (WO2020142557A1, compound 6).
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DescriptionMenin-MLL inhibitor 20 is an irreversible menin-MLL interaction inhibitor with antitumor activities (WO2020142557A1, compound 6).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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Recptorγ-secretase
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Research Area——
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Indication——
Chemical Information
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CAS Number2448173-47-3
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Formula Weight612.72
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Molecular FormulaC33H40N8O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 33.33 mg/mL (54.40 mM)
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SMILESCC(C)(C)OC(N[C@H]1CN(Cc2cc(C(Nc(cc3)ccc3-c([nH]3)cc4c3ncnc4N3CCOCC3)=O)ncc2)CCC1)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhao B, et al. Identification of gamma-secretase inhibitor potency determinants on presenilin. J Biol Chem. 2008 Feb 1;283(5):2927-38.
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