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IU1-248
CAS No. 2307472-03-1
IU1-248( —— )
Catalog No. M28642 CAS No. 2307472-03-1
IU1-248 is a derivative of IU1. IU1-248 is a potent and selective USP14 inhibitor with an IC50 of 0.83 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 104 | In Stock |
|
| 5MG | 93 | In Stock |
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| 10MG | 155 | In Stock |
|
| 25MG | 318 | In Stock |
|
| 50MG | 439 | In Stock |
|
| 100MG | 626 | In Stock |
|
| 200MG | 873 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameIU1-248
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NoteResearch use only, not for human use.
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Brief DescriptionIU1-248 is a derivative of IU1. IU1-248 is a potent and selective USP14 inhibitor with an IC50 of 0.83 μM.
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DescriptionIU1-248 is a derivative of IU1. IU1-248 is a potent and selective USP14 inhibitor with an IC50 of 0.83 μM.(In Vitro):IU1-248 exhibits an IC50 value of 0.83 μM toward USP14, which is 10-fold more potent than that of IU1 (IC50=12.25 μM).
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In VitroIU1-248 exhibits an IC50 value of 0.83?μM toward USP14, which is comparable to that of IU1-47 (IC50=0.68 μM) and 10-fold more potent than that of IU1 (IC50=12.25 μM).
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In Vivo——
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetDUB
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RecptorH1 receptor|Human Endogenous Metabolite|K+ current (IKr)|Cholinergic
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Research Area——
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Indication——
Chemical Information
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CAS Number2307472-03-1
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Formula Weight337.42
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Molecular FormulaC20H23N3O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 83.33 mg/mL (246.96 mM)
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SMILESCc1cc(C(CN(CC2)CCC2O)=O)c(C)n1-c(cc1)ccc1C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Sakuta H. Inhibition by histamine H1 receptor antagonists of endogenous glibenclamide-sensitive K+ channels in follicle-enclosed Xenopus oocytes. Eur J Pharmacol. 1994 Jan 1;266(1):99-102.
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