CVN424( —— )

Catalog No. M28619 CAS No. 2254706-21-1

CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	249	In Stock
5MG	236	In Stock
10MG	376	In Stock
25MG	620	In Stock
50MG	877	In Stock
100MG	1144	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

CVN424
Note

Research use only, not for human use.
Brief Description

CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.
Description

CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.(In Vivo): CVN424 is brain-penetrant and shows dose-dependent receptor occupancy that attained brain 50% of receptor occupancy at plasma concentrations of 6.0 and 7.4 ng/ml in mice and rats, respectively.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Cell Cycle/DNA Damage
Target

GPR
Recptor

5-HT4
Research Area

——
Indication

——

Chemical Information

CAS Number

2254706-21-1
Formula Weight

473.52
Molecular Formula

C24H29F2N5O3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 62.5 mg/mL (131.99 mM)
SMILES

CC(N(CC1)Cc(nc2N[C@H]3COCC3)c1nc2N(CC1)CCC1Oc(ccc(F)c1)c1F)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.R M Eglen, et al. Pharmacological characterization of two novel and potent 5-HT4 receptor agonists, RS 67333 and RS 67506, in vitro and in vivo. Br J Pharmacol. 1995 Aug;115(8):1387-92.

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