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TLR7/8/9-IN-1
CAS No. 2180127-82-4
TLR7/8/9-IN-1( —— )
Catalog No. M28232 CAS No. 2180127-82-4
TLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 169 | In Stock |
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| 2MG | 64 | In Stock |
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| 5MG | 113 | In Stock |
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| 10MG | 188 | In Stock |
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| 25MG | 307 | In Stock |
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| 50MG | 439 | In Stock |
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| 100MG | 597 | In Stock |
|
| 200MG | 853 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTLR7/8/9-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionTLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.
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DescriptionTLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayImmunology/Inflammation
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TargetTLR
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Recptor5-LOX
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Research Area——
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Indication——
Chemical Information
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CAS Number2180127-82-4
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Formula Weight435.6
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Molecular FormulaC27H37N3O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 83.33 mg/mL (191.30 mM)
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SMILESCC(C)c1c(-c(cc2)cc(OC)c2OC)[nH]c2c1cc(C1CCN(CCNC)CC1)cc2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Matthew Hutzler J, et al. In vitro-in vivo correlation and translation to the clinical outcome for CJ-13,610, a novel inhibitor of 5-lipoxygenase. Drug Metab Dispos. 2010 Jul;38(7):1113-21.
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