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A2A receptor antagonist 1
CAS No. 443103-97-7
A2A receptor antagonist 1( CPI-444 analog )
Catalog No. M28146 CAS No. 443103-97-7
A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 37 | In Stock |
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| 2MG | 33 | In Stock |
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| 5MG | 53 | In Stock |
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| 10MG | 85 | In Stock |
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| 25MG | 183 | In Stock |
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| 50MG | 274 | In Stock |
|
| 100MG | 407 | In Stock |
|
| 200MG | 578 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameA2A receptor antagonist 1
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NoteResearch use only, not for human use.
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Brief DescriptionA2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
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DescriptionA2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.(In Vitro):A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively.
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In VitroA2A receptor antagonist 1 (CPI-444 analog)?is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrates its binding activity with Ki values of 4 and 264 nM, respectively.
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In Vivo——
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SynonymsCPI-444 analog
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PathwayApoptosis
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TargetAdenosine Receptor
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RecptorMAGL
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Research Area——
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Indication——
Chemical Information
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CAS Number443103-97-7
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Formula Weight309.3
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Molecular FormulaC16H12FN5O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (80.83 mM)
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SMILESNc1nc(-c2ccco2)c2cnn(Cc3ccccc3F)c2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Aaltonen N, et al. Piperazine and piperidine triazole ureas as ultrapotent and highly selective inhibitors of monoacylglycerol lipase. Chem Biol. 2013 Mar 21;20(3):379-90.
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