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5-Benzyloxygramine
CAS No. 1453-97-0
5-Benzyloxygramine( —— )
Catalog No. M28056 CAS No. 1453-97-0
5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | 44 | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product Name5-Benzyloxygramine
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NoteResearch use only, not for human use.
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Brief Description5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
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Description5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.(In Vitro):5-Benzyloxygramine is a new N protein PPI orthosteric stabilizer that exhibits both antiviral and N-NTD protein-stabilizing activities. 5-benzyloxygramine stabilizes the N-NTD dimers through simultaneous hydrophobic interactions with both partners, resulting in abnormal N protein oligomerization that was further confirmed in the cell.
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In Vitro5-benzyloxygramine stabilizes the N-NTD dimers through simultaneous hydrophobic interactions with both partners, resulting in abnormal N protein oligomerization that was further confirmed in the cell.
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorAQP1
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Research Area——
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Indication——
Chemical Information
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CAS Number1453-97-0
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Formula Weight280.371
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Molecular FormulaC18H20N2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (891.71 mM)
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SMILESCN(C)Cc1c[nH]c2ccc(OCc3ccccc3)cc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Seeliger D, et al. Discovery of novel human aquaporin-1 blockers. ACS Chem Biol. 2013 Jan 18;8(1):249-56.
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