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MK-2295

CAS No. 878811-00-8

MK-2295( MK2295 | MK 2295 )

Catalog No. M27996 CAS No. 878811-00-8

MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	149	In Stock
10MG	220	In Stock
25MG	337	In Stock
50MG	462	In Stock
100MG	619	In Stock
200MG	835	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

MK-2295
Note

Research use only, not for human use.
Brief Description

MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
Description

MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
In Vitro

——
In Vivo

——
Synonyms

MK2295 | MK 2295
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

JAK1
Research Area

——
Indication

——

Chemical Information

CAS Number

878811-00-8
Formula Weight

490.583
Molecular Formula

C27H31FN6O2
Purity

>98% (HPLC)
Solubility

——
SMILES

C[C@@H]1CCCN1c1nc(cc(n1)-c1ccc(F)cc1)N1CCN(C[C@H]1C)c1ncc(cc1C)C(O)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Paul Smith, et al. Use of jak1 inhibitors for the treatment of cutaneous lupus erythematosus and lichen planus (lp). WO2021076124A1.

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