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Home - Products - Metabolic Enzyme/Protease - PAI-1 - Aleplasinin

Aleplasinin

CAS No. 481629-87-2

Aleplasinin( PAZ-417 | PAZ 417 | PAZ417 )

Catalog No. M27948 CAS No. 481629-87-2

Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Aleplasinin
  • Note
    Research use only, not for human use.
  • Brief Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PAZ-417 | PAZ 417 | PAZ417
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    PAI-1
  • Recptor
    nAChR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    481629-87-2
  • Formula Weight
    425.528
  • Molecular Formula
    C28H27NO3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (587.52 mM)
  • SMILES
    Cc1cccc(c1)-c1ccc2n(Cc3ccc(cc3)C(C)(C)C)cc(C(=O)C(O)=O)c2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kimura I, et al. Inotropic effects of (+/-)-higenamine and its chemically related components, (+)-R-coclaurine and (+)-S-reticuline, contained in the traditional sino-Japanese medicines "bushi" and "shin-i" in isolated guinea pig papillary muscle. Jpn J Pharmacol. 1989 May;50(1):75-8.
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