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Suprafenacine
CAS No. 1477482-50-0
Suprafenacine( N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide )
Catalog No. M27928 CAS No. 1477482-50-0
Suprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 129 | In Stock |
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| 2MG | 78 | In Stock |
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| 5MG | 126 | In Stock |
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| 10MG | 179 | In Stock |
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| 25MG | 321 | In Stock |
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| 50MG | 442 | In Stock |
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| 100MG | 625 | In Stock |
|
| 200MG | 826 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameSuprafenacine
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NoteResearch use only, not for human use.
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Brief DescriptionSuprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase.
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DescriptionSuprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase. Suprafenacine binds to microtubules and inhibits aggregation at the colchicine junction. Suprafenacine is selective for cancer cells, including drug-resistant cancer cells.
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In Vitro——
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In Vivo——
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SynonymsN'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetMicrotubule/Tubulin
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Recptorβ2-adrenergic receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1477482-50-0
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Formula Weight282.347
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Molecular FormulaC16H18N4O
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Purity>98% (HPLC)
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Solubility——
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SMILESCc1ccc(\C=N\NC(=O)c2n[nH]c3CCCCc23)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Shuyun Bi, et al. Study on the interactions of mapenterol with serum albumins using multi-spectroscopy and molecular docking. Luminescence. 2016 Mar;31(2):372-379.
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