Adaptaquin
CAS No. 385786-48-1
Adaptaquin( —— )
Catalog No. M27498 CAS No. 385786-48-1
Adaptaquin is an inhibitor of the hypoxia-inducing factor prolyl hydroxylase (HIF-PH).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 5MG | 28 | In Stock |
|
| 10MG | 46 | In Stock |
|
| 25MG | 93 | In Stock |
|
| 50MG | 147 | In Stock |
|
| 100MG | 231 | In Stock |
|
| 200MG | 328 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameAdaptaquin
-
NoteResearch use only, not for human use.
-
Brief DescriptionAdaptaquin is an inhibitor of the hypoxia-inducing factor prolyl hydroxylase (HIF-PH).
-
DescriptionAdaptaquin is an inhibitor of the hypoxia-inducing factor prolyl hydroxylase (HIF-PH).
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayAngiogenesis
-
TargetHIF/HIF Prolyl-hydroxylase
-
RecptorNEK6
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number385786-48-1
-
Formula Weight377.82
-
Molecular FormulaC21H16ClN3O2
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 100 mg/mL (264.68 mM)
-
SMILESOc1cccnc1NC(c(cc1)ccc1Cl)c(ccc1cccnc11)c1O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.De Donato M, et al. Identification and antitumor activity of a novel inhibitor of the NIMA-related kinase NEK6. Sci Rep. 2018;8(1):16047. Published 2018 Oct 30.
molnova catalog
related products
-
ZINC13466751
ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 μM).
-
HIF-IN-1
HIF-IN-1 is a potent inhibitor of hypoxia-inducible factor (HIF-1), which is associated with tumor and cancer cell proliferation and inhibits HIF-1α protein aggregation.
-
Molidustat
Molidustat (BAY 85-3934) is an orally active small molecule inhibitor of hypoxia inducible factor prolyl hydroxylase (HIF-PH) with IC50 of 480 nM, 280 nM and 450 nM for PHD1, PHD2, and PHD3, respectively.
Cart
sales@molnova.com