BD 1008 dihydrobromide

CAS No. 138356-09-9

BD 1008 dihydrobromide( —— )

Catalog No. M27463 CAS No. 138356-09-9

BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 69 In Stock
2MG 33 In Stock
5MG 53 In Stock
10MG 93 In Stock
25MG 227 In Stock
50MG 347 In Stock
100MG 494 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    BD 1008 dihydrobromide
  • Note
    Research use only, not for human use.
  • Brief Description
    BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM).
  • Description
    BD1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. BD1008 dihydrobromide attenuate the toxicity and stimulant effects of cocaine through antagonism of sigma receptors.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Autophagy
  • Target
    Sigma receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    138356-09-9
  • Formula Weight
    463.08
  • Molecular Formula
    C15H24Br2Cl2N2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Br.Br.CN(CCN1CCCC1)CCc1ccc(Cl)c(Cl)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Barakat MT, et al. Simethicone is retained in endoscopes despite reprocessing: impact of its use on working channel fluid retention and adenosine triphosphate bioluminescence values (with video). Gastrointest Endosc. 2018 Aug 17.
molnova catalog
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