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Lp-PLA2-IN-1

CAS No. 1420367-28-7

Lp-PLA2-IN-1( Lp-PLA2 -IN-1 | Lp-PLA2 inhibitor 1 )

Catalog No. M26743 CAS No. 1420367-28-7

Lp-PLA2 -IN-1 suppresses Lp-PLA2 activity processes for their preparation.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Lp-PLA2-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    Lp-PLA2 -IN-1 suppresses Lp-PLA2 activity processes for their preparation.
  • Description
    Lp-PLA2 -IN-1 suppresses Lp-PLA2 activity processes for their preparation. Lp-PLA2 -IN-1also inhibits to compositions containing them and to their use in the treatment of diseases associated with the activity of Lp-PLA2, for example, atherosclerosis, Alzheimer's disease.(In Vitro):Lp-PLA2 is a phospholipase A2 enzyme involved in the hydrolysis of lipoprotein lipids or phospholipids. Lp-PLA2 travels with LDL and rapidly cleaves oxidized phosphatidylcholine molecules derived from the oxidation of LDL.
  • In Vitro
    Lipoprotein-associated phospholipase A2 (Lp-PLA2) is a phospholipase A2 enzyme involved in hydrolysis of lipoprotein lipids or phospholipids. Lp-PLA2 travels with low-density lipoprotein (LDL) and rapidly cleaves oxidized phosphatidylcholine molecules derived from the oxidation of LDL.
  • In Vivo
    ——
  • Synonyms
    Lp-PLA2 -IN-1 | Lp-PLA2 inhibitor 1
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phospholipase
  • Recptor
    Androgen Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1420367-28-7
  • Formula Weight
    468.384
  • Molecular Formula
    C21H17F5N4O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?Ethanol : 25 mg/mL (53.38 mM)
  • SMILES
    CN1CCCn2c1cc(OCc1cc(F)c(Oc3ccc(nc3)C(F)(F)F)c(F)c1)nc2=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cutler C, et al. Equine metabolism of the selective androgen receptor modulator AC-262536 in vitro and in urine, plasma and hair following oral administration. Drug Test Anal. 2021 Feb;13(2):369-385.
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