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Entasobulin

CAS No. 501921-61-5

Entasobulin( —— )

Catalog No. M26678 CAS No. 501921-61-5

Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 40 In Stock
5MG 36 In Stock
10MG 55 In Stock
25MG 93 In Stock
50MG 161 In Stock
100MG 254 In Stock
200MG 365 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Entasobulin
  • Note
    Research use only, not for human use.
  • Brief Description
    Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.
  • Description
    Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.(In Vitro):Entasobulin is an indolizine-glyoxylamide based small molecule. It shows substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
  • In Vitro
    Entasobulin is a indolizine-glyoxylamide based small molecule that demonstrate substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Microtubule/Tubulin
  • Recptor
    MLLT1| MLLT3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    501921-61-5
  • Formula Weight
    439.9
  • Molecular Formula
    C26H18ClN3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 155 mg/mL (352.36 mM)
  • SMILES
    Clc1ccc(Cn2cc(C(=O)C(=O)Nc3ccc4ncccc4c3)c3ccccc23)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Moustakim M, et al. Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Angew Chem Int Ed Engl. 2018 Dec 10;57(50):16302-16307.
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