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Entasobulin
CAS No. 501921-61-5
Entasobulin( —— )
Catalog No. M26678 CAS No. 501921-61-5
Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 40 | In Stock |
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| 5MG | 36 | In Stock |
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| 10MG | 55 | In Stock |
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| 25MG | 93 | In Stock |
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| 50MG | 161 | In Stock |
|
| 100MG | 254 | In Stock |
|
| 200MG | 365 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEntasobulin
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NoteResearch use only, not for human use.
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Brief DescriptionEntasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.
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DescriptionEntasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.(In Vitro):Entasobulin is an indolizine-glyoxylamide based small molecule. It shows substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
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In VitroEntasobulin is a indolizine-glyoxylamide based small molecule that demonstrate substantial in vitro anti-proliferative activities against cancer cell lines, including multidrug resistance (MDR) phenotypes.
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In Vivo——
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetMicrotubule/Tubulin
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RecptorMLLT1| MLLT3
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Research Area——
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Indication——
Chemical Information
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CAS Number501921-61-5
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Formula Weight439.9
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Molecular FormulaC26H18ClN3O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 155 mg/mL (352.36 mM)
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SMILESClc1ccc(Cn2cc(C(=O)C(=O)Nc3ccc4ncccc4c3)c3ccccc23)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Moustakim M, et al. Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Angew Chem Int Ed Engl. 2018 Dec 10;57(50):16302-16307.
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