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DGAT1-IN-1
CAS No. 1449779-49-0
DGAT1-IN-1( —— )
Catalog No. M26665 CAS No. 1449779-49-0
DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 141 | In Stock |
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| 2MG | 75 | In Stock |
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| 5MG | 116 | In Stock |
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| 10MG | 187 | In Stock |
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| 25MG | 359 | In Stock |
|
| 50MG | 529 | In Stock |
|
| 100MG | 762 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDGAT1-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionDGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).
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DescriptionDGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).(In Vitro):Various concentrations (0.0008 μΜ, 0.004 μΜ, 0.02 μΜ, 0.1 μΜ, 0.5 μΜ, 2.5 μΜ and 10.0 μΜ) of the compounds of Examples were added to individual wells prior to the addition of the cell lysates, or human or mouse liver microsomes.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetTransferase
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RecptorCentromere-Associated Protein E
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Research Area——
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Indication——
Chemical Information
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CAS Number1449779-49-0
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Formula Weight551.566
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Molecular FormulaC30H28F3N3O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 20 mg/mL (36.26 mM)
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SMILESOC(=O)C[C@H]1CC[C@@H](CC1)c1ccc(cc1)-c1ccc2nc(cn2c1)C(=O)NCc1ccc(OC(F)(F)F)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Qian X, et al. Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. ACS Med Chem Lett. 2010 Jan 19;1(1):30-4.
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