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CRAC intermediate 1
CAS No. 1249343-86-9
CRAC intermediate 1( 5-(S)-Fluorowillardiine )
Catalog No. M26129 CAS No. 1249343-86-9
CRAC intermediate 1 is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 10MG | 31 | In Stock |
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| 25MG | 59 | In Stock |
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| 50MG | 91 | In Stock |
|
| 100MG | 138 | In Stock |
|
| 200MG | 206 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCRAC intermediate 1
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NoteResearch use only, not for human use.
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Brief DescriptionCRAC intermediate 1 is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
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DescriptionCRAC intermediate 1 is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
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In Vitro——
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In Vivo——
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Synonyms5-(S)-Fluorowillardiine
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorAMPA
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Research Area——
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Indication——
Chemical Information
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CAS Number1249343-86-9
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Formula Weight223.183
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Molecular FormulaC10H7F2N3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 50 mg/mL (224.03 mM)
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SMILESFc1cccc(F)c1C(=O)Nc1cc[nH]n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Arai AC, Kessler M, Rogers G, Lynch G. Effects of the potent ampakine CX614 on hippocampal and recombinant AMPA receptors: interactions with cyclothiazide and GYKI 52466. Mol Pharmacol. 2000 Oct;58(4):802-13. PubMed PMID: 10999951.
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