G-1

CAS No. 881639-98-1

G-1( —— )

Catalog No. M24897 CAS No. 881639-98-1

G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 71 In Stock
5MG 73 In Stock
10MG 117 In Stock
25MG 202 In Stock
50MG 314 In Stock
100MG 454 In Stock
200MG 649 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    G-1
  • Note
    Research use only, not for human use.
  • Brief Description
    G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
  • Description
    G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    GPR30
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    881639-98-1
  • Formula Weight
    412.28
  • Molecular Formula
    C21H18BrNO3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:50 mg/mL (121.28 mM; Need ultrasonic);H2O:< 0.1 mg/mL (insoluble)
  • SMILES
    CC(=O)C1=CC2=C(C=C1)NC(C3C2C=CC3)C4=CC5=C(C=C4Br)OCO5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cheng Q, et al. G-1 exerts neuroprotective effects through G protein-coupled estrogen receptor 1 following spinal cord injury in mice. Biosci Rep. 2016 Aug 31;36(4). pii: e00373.
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