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Vanilloid receptor antagonist 1

CAS No. 871814-52-7

Vanilloid receptor antagonist 1( 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile )

Catalog No. M24886 CAS No. 871814-52-7

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	37	In Stock
5MG	235	In Stock
10MG	353	In Stock
25MG	601	In Stock
50MG	830	In Stock
100MG	1181	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Vanilloid receptor antagonist 1
Note

Research use only, not for human use.
Brief Description

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
Description

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
In Vitro

——
In Vivo

——
Synonyms

4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

TRPV1
Research Area

——
Indication

——

Chemical Information

CAS Number

871814-52-7
Formula Weight

305.33
Molecular Formula

C18H15N3O2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (327.51 mM)
SMILES

CC(C)C(N1c(cc2)ccc2C#N)=Nc(cc(cc2)O)c2C1=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Ritchie T J , Culshaw A J , Brain C T , et al. Quinazolinone derivatives useful as vanilloid antagonists: US, US8349852 B2[P]. 2012.

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