BIM-46187 4HCl

CAS No. 2489449-03-6

BIM-46187 4HCl( PH-064 4HCl )

Catalog No. M24135 CAS No. 2489449-03-6

PH-064 4HCl is a heterotrimeric G-protein complex inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 178 In Stock
5MG 268 In Stock
10MG 399 In Stock
25MG 659 In Stock
50MG 888 In Stock
100MG 1251 In Stock
500MG 2511 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    BIM-46187 4HCl
  • Note
    Research use only, not for human use.
  • Brief Description
    PH-064 4HCl is a heterotrimeric G-protein complex inhibitor.
  • Description
    PH-064 4HCl is a heterotrimeric G-protein complex inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PH-064 4HCl
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    heterotrimeric G-protein complex
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2489449-03-6
  • Formula Weight
    940.95
  • Molecular Formula
    C44H62Cl4N8O2S2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    O=C([C@@H](N)CSSC[C@H](N)C(N(CCN1C2=NC(C3=CC=CC=C3)=C1)[C@H]2CC4CCCCC4)=O)N5[C@H](C6=NC(C7=CC=CC=C7)=CN6CC5)CC8CCCCC8.Cl.Cl.Cl.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Favre-Guilmard C, et al. The novel inhibitor of the heterotrimeric G-protein complex, BIM-46187, elicits anti-hyperalgesic properties and synergizes with morphine. Eur J Pharmacol. 2008 Oct 10;594(1-3):70-6.
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