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NVP-BHG712 isomer
CAS No. 2245892-85-5
NVP-BHG712 isomer( —— )
Catalog No. M24025 CAS No. 2245892-85-5
NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 46 | In Stock |
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| 5MG | 72 | In Stock |
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| 10MG | 138 | In Stock |
|
| 25MG | 246 | In Stock |
|
| 50MG | 356 | In Stock |
|
| 100MG | 530 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameNVP-BHG712 isomer
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NoteResearch use only, not for human use.
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Brief DescriptionNVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
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DescriptionNVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
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In VitroNVP-BHG712 isomer exhibits IC 50 values of 163 nM and 1660 nM for EPHA2 and EPHA4, respectively.
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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TargetEphrin Receptor
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RecptorEPHA2
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Research Area——
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Indication——
Chemical Information
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CAS Number2245892-85-5
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Formula Weight503.48
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Molecular FormulaC26H20F3N7O
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL (99.31 mM; Need ultrasonic);H2O:insoluble
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SMILESO=C(NC1=CC=CC(C(F)(F)F)=C1)C2=CC=C(C)C(NC3=NC(C4=CC=CN=C4)=NC5=NN(C)C=C53)=C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tr?ster A, et al. NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family. ChemMedChem. 2018 Aug 20;13(16):1629-1633.
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