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SBI-553
CAS No. 1849603-72-0
SBI-553( —— )
Catalog No. M23841 CAS No. 1849603-72-0
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 102 | In Stock |
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| 5MG | 92 | In Stock |
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| 10MG | 169 | In Stock |
|
| 25MG | 353 | In Stock |
|
| 50MG | 555 | In Stock |
|
| 100MG | 888 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSBI-553
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NoteResearch use only, not for human use.
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Brief DescriptionSBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
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DescriptionSBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetNeurotensin Receptor
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RecptorNTR1
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Research Area——
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Indication——
Chemical Information
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CAS Number1849603-72-0
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Formula Weight450.55
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Molecular FormulaC26H31FN4O2
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Purity>98% (HPLC)
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SolubilityDMSO:62.5 mg/mL (138.72 mM; Need ultrasonic)
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SMILESCN(CCO)C1=CC2=C(C=C1)N=C(N=C2N3CCC(CC3)C4=CC=CC=C4OC)C5(CC5)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Pinkerton AB, et al. Discovery of β-Arrestin Biased, Orally Bioavailable, and CNS Penetrant Neurotensin Receptor 1 (NTR1) Allosteric Modulators. J Med Chem. 2019 Aug 20.
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