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Cav 2.2 blocker 1

CAS No. 1567335-29-8

Cav 2.2 blocker 1( —— )

Catalog No. M23678 CAS No. 1567335-29-8

Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 113 In Stock
5MG 107 In Stock
10MG 183 In Stock
25MG 340 In Stock
50MG 510 In Stock
100MG 764 In Stock
200MG 1004 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Cav 2.2 blocker 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
  • Description
    Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Cav 2.2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1567335-29-8
  • Formula Weight
    424.96
  • Molecular Formula
    C25H29ClN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:20 mg/mL (47.07 mM; Need ultrasonic)
  • SMILES
    CC1(C)CC(C2=NN(C3=CC=CC=C3OC)C(C4=CC=C(Cl)C=C4)=C2)CC(C)(C)O1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Wall MJ, et al. Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment of pain. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3780-3783.
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