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Cav 2.2 blocker 1

CAS No. 1567335-29-8

Cav 2.2 blocker 1( —— )

Catalog No. M23678 CAS No. 1567335-29-8

Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Cav 2.2 blocker 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
  • Description
    Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Cav 2.2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1567335-29-8
  • Formula Weight
    424.96
  • Molecular Formula
    C25H29ClN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:20 mg/mL (47.07 mM; Need ultrasonic)
  • SMILES
    CC1(C)CC(C2=NN(C3=CC=CC=C3OC)C(C4=CC=C(Cl)C=C4)=C2)CC(C)(C)O1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Wall MJ, et al. Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment of pain. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3780-3783.
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