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PROTAC ERRα ligand 1
CAS No. 1264754-13-3
PROTAC ERRα ligand 1( —— )
Catalog No. M23437 CAS No. 1264754-13-3
PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 66 | In Stock |
|
| 2MG | 35 | In Stock |
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| 5MG | 55 | In Stock |
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| 10MG | 84 | In Stock |
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| 25MG | 149 | In Stock |
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| 50MG | 238 | In Stock |
|
| 100MG | 356 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 764 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePROTAC ERRα ligand 1
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NoteResearch use only, not for human use.
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Brief DescriptionPROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
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DescriptionPROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorERRα|ERRγ
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Research Area——
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Indication——
Chemical Information
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CAS Number1264754-13-3
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Formula Weight420.36
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Molecular FormulaC19H11F3N2O4S
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Purity>98% (HPLC)
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SolubilityDMSO : 120 mg/mL (285.47 mM; Need ultrasonic)
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SMILESN#CC1=CC=C(OC2=CC=C(/C=C(SC(N3)=O)/C3=O)C=C2OC)C(C(F)(F)F)=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Patch RJ, et al. Identification of diaryl ether-based ligands for estrogen-related receptor α as potential antidiabetic agents. J Med Chem. 2011 Feb 10;54(3):788-808.
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