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HA-155
CAS No. 1229652-22-5
HA-155( Autotaxin Inhibitor IV )
Catalog No. M23406 CAS No. 1229652-22-5
HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 93 | In Stock |
|
| 10MG | 148 | In Stock |
|
| 25MG | 310 | In Stock |
|
| 50MG | 454 | In Stock |
|
| 100MG | 639 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameHA-155
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NoteResearch use only, not for human use.
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Brief DescriptionHA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
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DescriptionHA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
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In Vitro——
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In Vivo——
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SynonymsAutotaxin Inhibitor IV
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PathwayAngiogenesis
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TargetPDE
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RecptorATX (autotaxin)
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Research Area——
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Indication——
Chemical Information
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CAS Number1229652-22-5
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Formula Weight463.29
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Molecular FormulaC24H19BFNO5S
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESB(C1=CC=C(C=C1)COC2=CC=C(C=C2)/C=C\3/C(=O)N(C(=O)S3)CC4=CC=C(C=C4)F)(O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Albers H M H G , Hendrickx L J D , Van Tol R J P , et al. Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin[J]. Journal of Medicinal Chemistry, 2011, 54(13):4619-26.
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