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DPCPX
CAS No. 102146-07-6
DPCPX( PD 116948 )
Catalog No. M23228 CAS No. 102146-07-6
DPCPX is an A1 adenosine receptor antagonist
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 43 | In Stock |
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| 5MG | 29 | In Stock |
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| 10MG | 39 | In Stock |
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| 25MG | 62 | In Stock |
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| 50MG | 91 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDPCPX
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NoteResearch use only, not for human use.
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Brief DescriptionDPCPX is an A1 adenosine receptor antagonist
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DescriptionDPCPX is an A1 adenosine receptor antagonist.
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In Vitro——
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In VivoDPCPX (PD 116948) ( 0.1, 0.3 and 1.0 mg/kg i.v. ) produces significant dose-related increases (P<0.05) in urine volume and in urinary sodium, potassium and chloride excretion.
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SynonymsPD 116948
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PathwayApoptosis
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TargetAdenosine Receptor
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RecptorA1
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Research Area——
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Indication——
Chemical Information
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CAS Number102146-07-6
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Formula Weight304.39
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Molecular FormulaC16H24N4O2
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Purity>98% (HPLC)
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SolubilityDMSO:<1 mg/mL;Ethanol:<1 mg/mL
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SMILESCCCN(c1c(C(N2CCC)=O)[nH]c(C3CCCC3)n1)C2=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Aleksandra S , Ewa P , Karolina B , et al. DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests[J]. Naunyn-Schmiedeberg's Archives of Pharmacology, 2018:1-11.
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