Leuphasyl TFA
CAS No. 67586-27-0
Leuphasyl TFA( —— )
Catalog No. M22894 CAS No. 67586-27-0
Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 107 | In Stock |
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| 5MG | 172 | In Stock |
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| 10MG | 258 | In Stock |
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| 25MG | 426 | In Stock |
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| 50MG | 586 | In Stock |
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| 100MG | 792 | In Stock |
|
| 200MG | 1051 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLeuphasyl TFA
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NoteResearch use only, not for human use.
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Brief DescriptionLeuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors.
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DescriptionLeuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors. Leuphasyl TFA is a potent, long-acting Leu-enkephalin analog that is resistant to enzymatic degradation.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptorδ-opioid receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number67586-27-0
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Formula Weight683.67
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Molecular FormulaC31H40F3N5O9
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Purity>98% (HPLC)
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Solubility——
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SMILESOc2ccc(C[C@H](N)C(=O)N[C@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)O)cc2.FC(F)(F)C(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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UFP-101
Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors. Antinociceptive and opposes the action of nociceptin in vivo.
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Endomorphin 2?
Endomorphins-2 (EM-2) could decrease both the frequency and amplitude of the sEPSC of the motoneurons in lamina IX which was reversed by the MOR antagonist CTOP.??
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Spinorphin
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.Spinorphin inhibited cytoplasmic Ca(2+) ([Ca(2+)]i) transients, evoked by depolarization and capsaicin selectively in medium and small cultured rat DRG neurons.?
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