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9-FLUORENOL
CAS No. 1689-64-1
9-FLUORENOL( —— )
Catalog No. M22199 CAS No. 1689-64-1
9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | 27 | In Stock |
|
Biological Information
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Product Name9-FLUORENOL
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NoteResearch use only, not for human use.
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Brief Description9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.
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Description9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Fluorenol(100 mg/kg) is reported to promote wakefulness in mice with 39% increased effectiveness over the structurally related compound, modafinil.
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In Vitro——
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In VivoPharmacokinetic parameters of 9-Fluorenol (100 mg/kg; i.p.) in rats
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Synonyms——
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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Recptordopamine reuptake
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Research Area——
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Indication——
Chemical Information
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CAS Number1689-64-1
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Formula Weight182.22
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Molecular FormulaC13H10O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (548.79 mM)
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SMILESOC2([H])c1ccccc1c3ccccc23
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Dunn D , Hostetler G , Iqbal M , et al. Wake promoting agents: Search for next generation modafinil, lessons learned: Part III[J]. Bioorganic & Medicinal Chemistry Letters, 2012, 22(11):3751-3753.
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