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(E/Z)-GSK5182?

CAS No. ——

(E/Z)-GSK5182?( GSK5182(Z/E) )

Catalog No. M22036 CAS No. ——

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

(E/Z)-GSK5182?
Note

Research use only, not for human use.
Brief Description

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers.
Description

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active estrogen-related receptor γ (ERRγ) inverse agonist(IC50 of 79 nM),and also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma.
In Vitro

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In Vivo

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Synonyms

GSK5182(Z/E)
Pathway

Endocrinology/Hormones
Target

Estrogen Receptor/ERR
Recptor

ERRγ|ROS
Research Area

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Indication

——

Chemical Information

CAS Number

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Formula Weight

417.54
Molecular Formula

C27H31NO3
Purity

>98% (HPLC)
Solubility

DMSO:95 mg/mL?(227.52 mM;?Need ultrasonic)
SMILES

CN(C)CCOC1=CC=C(C=C1)C(=C(CCCO)C1=CC=CC=C1)C1=CC=C(O)C=C1
Chemical Name

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Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Misra J, et al. ERRγ: a Junior Orphan with a Senior Role in Metabolism. Trends Endocrinol Metab. 2017 Apr;28(4):261-272.

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