Oncrasin 1

CAS No. 75629-57-1

Oncrasin 1( —— )

Catalog No. M21162 CAS No. 75629-57-1

Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 62 In Stock
5MG 29 In Stock
10MG 37 In Stock
25MG 56 In Stock
50MG 102 In Stock
100MG 189 In Stock
200MG 272 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Oncrasin 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations.
  • Description
    Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    Ras
  • Recptor
    K-Ras
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    75629-57-1
  • Formula Weight
    269.73
  • Molecular Formula
    C16H12ClNO
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:43 mg/mL (159.42 mM)
  • SMILES
    O=Cc1cn(Cc2ccc(Cl)cc2)c2ccccc12
  • Chemical Name
    1-(4-Chlorobenzyl)-1H-indole-3-carbaldehyde

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Guo W Wu S Liu J et al. Identification of a Small Molecule with Synthetic Lethality for K-Ras and Protein Kinase C Iota[J]. Cancer Research 2008 68(18):7403-7408.
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