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VPS34 inhibitor 1 (Compound 19 PIK-III analogue)
CAS No. 1383716-46-8
VPS34 inhibitor 1 (Compound 19 PIK-III analogue)( PIK-III analogue )
Catalog No. M21136 CAS No. 1383716-46-8
VPS34 inhibitor 1 (Compound 19 PIK-III analogue) is a potent and selective inhibitor of VPS34( IC50 : 15 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 154 | In Stock |
|
| 5MG | 140 | In Stock |
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| 10MG | 227 | In Stock |
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| 25MG | 398 | In Stock |
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| 50MG | 554 | In Stock |
|
| 100MG | 737 | In Stock |
|
| 200MG | 1014 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVPS34 inhibitor 1 (Compound 19 PIK-III analogue)
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NoteResearch use only, not for human use.
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Brief DescriptionVPS34 inhibitor 1 (Compound 19 PIK-III analogue) is a potent and selective inhibitor of VPS34( IC50 : 15 nM).
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DescriptionVPS34 inhibitor 1 (Compound 19 PIK-III analogue) is a potent and selective inhibitor of VPS34( IC50 : 15 nM).
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In Vitro——
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In Vivo——
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SynonymsPIK-III analogue
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorVps34
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Research Area——
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Indication——
Chemical Information
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CAS Number1383716-46-8
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Formula Weight391.47
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Molecular FormulaC21H25N7O
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Purity>98% (HPLC)
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SolubilityDMSO:78 mg/mL (199.25 mM)
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SMILESCC(C)(O)CNc1ncc(-c2ccnc(Nc3ccncc3)n2)c(CC2CC2)n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Honda A Harrington E Cornella-Taracido I et al. Potent Selective and Orally Bioavailable Inhibitors of VPS34 Provide Chemical Tools to Modulate Autophagy in Vivo[J]. ACS Medicinal Chemistry Letters 2015 7(1).
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