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Deltorphin I(TFA)
CAS No. 122752-15-2
Deltorphin I(TFA)( Deltorphin 1 | Deltorphin C )
Catalog No. M21043 CAS No. 122752-15-2
Deltorphin I(TFA) is an agonist of δ-opioid receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 206 | In Stock |
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| 5MG | 140 | In Stock |
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| 10MG | 211 | In Stock |
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| 25MG | 356 | In Stock |
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| 50MG | 513 | In Stock |
|
| 100MG | 732 | In Stock |
|
| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameDeltorphin I(TFA)
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NoteResearch use only, not for human use.
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Brief DescriptionDeltorphin I(TFA) is an agonist of δ-opioid receptor.
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DescriptionDeltorphin I(TFA) is an agonist of δ-opioid receptor.
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In Vitro——
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In VivoTwice daily administration of Deltorphin I (20μg/mouse) for 4 days produces tolerance to Deltorphin I analgesia, as shown by the decrease in the analgesic response. The peak analgesic response to Deltorphin I (20 μg/mouse) at 10 min after injections is decreased from 8.36±0.28 s (the 1st day) to 4.53±0.14 s (the 4th day) markedly. Concurrent treatment of Melatonin (0.5, 1 and 2.5 mg/kg) and Deltorphin I (20 μg/mouse) twice daily for 4 days can attenuate the tolerance to Deltorphin I analgesia (P<0.05, <0.05 and <0.05), and this effect is dose dependent.
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SynonymsDeltorphin 1 | Deltorphin C
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptorδ-opioid receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number122752-15-2
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Formula Weight768.86
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Molecular FormulaC37H52N8O10
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (32.52 mM)
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SMILESCC(C)[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)NCC(N)=O)C(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Dupin S Tafani J A M Honoré Mazarguil et al. [125I][D-Ala2]deltorphin-I: A high affinity delta-selective opioid receptor ligand[J]. Peptides 1991 12(4):825-830.
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