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Lixivaptan
CAS No. 168079-32-1
Lixivaptan( VPA-985 | WAY-VPA 985 )
Catalog No. M20804 CAS No. 168079-32-1
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 47 | In Stock |
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| 5MG | 67 | In Stock |
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| 10MG | 116 | In Stock |
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| 25MG | 236 | In Stock |
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| 50MG | 401 | In Stock |
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| 100MG | 591 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLixivaptan
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NoteResearch use only, not for human use.
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Brief DescriptionLixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM).
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DescriptionLixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM).
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In Vitro——
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In Vivo——
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SynonymsVPA-985 | WAY-VPA 985
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PathwayGPCR/G Protein
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TargetVasopressin Receptor
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RecptorVasopressin Receptor
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Research AreaMetabolic Disease
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IndicationAutosomal dominant polycystic kidney disease
Chemical Information
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CAS Number168079-32-1
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Formula Weight473.93
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Molecular FormulaC27H21ClFN3O2
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Purity>98% (HPLC)
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SolubilityDMSO:150 mg/mL (316.50 mM)
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SMILESCc1ccc(F)cc1C(=O)Nc1ccc(C(=O)N2Cc3cccn3Cc3ccccc32)c(Cl)c1
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Chemical NameN-(3-chloro-4-(1011-dihydro-6H-benzo[e]pyrrolo[12-a][14]diazepine-5-carbonyl)phenyl)-5-fluoro-2-methylbenzamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Wang X Constans MM Chebib FT.et al.Effect of a Vasopressin V2 Receptor Antagonist on Polycystic Kidney Disease Development in a Rat Model[J].Am J Nephrol. 2019;49(6):487-493.
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