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ONC212
CAS No. 1807861-48-8
ONC212( —— )
Catalog No. M20724 CAS No. 1807861-48-8
ONC212 a fluorinated-ONC201 analogue is a selective agonist of GPR132.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 92 | In Stock |
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| 5MG | 93 | In Stock |
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| 10MG | 154 | In Stock |
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| 25MG | 261 | In Stock |
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| 50MG | 410 | In Stock |
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| 100MG | 604 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameONC212
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NoteResearch use only, not for human use.
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Brief DescriptionONC212 a fluorinated-ONC201 analogue is a selective agonist of GPR132.
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DescriptionONC212 a fluorinated-ONC201 analogue is a selective agonist of GPR132.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetGHSR
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RecptorGPR132
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Research Area——
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Indication——
Chemical Information
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CAS Number1807861-48-8
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Formula Weight440.46
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Molecular FormulaC24H23F3N4O
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL (113.52 mM)
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SMILESFC(F)(F)c1ccc(CN2C3=NCCN3C3=C(CN(Cc4ccccc4)CC3)C2=O)cc1
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Chemical Name246789-Hexahydro-7-(phenylmethyl)-4-[[4-(trifluoromethyl)phenyl]methyl]imidazo[12-a]pyrido[34-e]pyrimidin-5(1H)-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Nii T Prabhu VV Ruvolo Vet al.Imipridone ONC212 activates orphan G protein-coupled receptor GPR132 and integrated stress response in acute myeloid leukemia[J].Leukemia. 2019 Dec;33(12):2805-2816.
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