Dimethylfraxetin

CAS No. 6035-49-0

Dimethylfraxetin( 678-Trimethoxycoumarin | Fraxetin dimethyl ether )

Catalog No. M20278 CAS No. 6035-49-0

Dimethylfraxetin is a Carbonic anhydrase inhibitor(Ki:0.0097 μM)

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 89 In Stock
5MG 72 In Stock
10MG 129 In Stock
25MG 259 In Stock
50MG 365 In Stock
100MG 514 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Dimethylfraxetin
  • Note
    Research use only, not for human use.
  • Brief Description
    Dimethylfraxetin is a Carbonic anhydrase inhibitor(Ki:0.0097 μM)
  • Description
    Dimethylfraxetin is a Carbonic anhydrase inhibitor.(Ki:0.0097 μM).
  • In Vitro
    At CA I there is one stand out compound being Dimethylfraxetin (compound 17), a nanomolar CA I inhibitor. This trimethoxy coumarin is the most potent of any of the NP coumarins across the six CA isozymes of the present study.
  • In Vivo
    ——
  • Synonyms
    678-Trimethoxycoumarin | Fraxetin dimethyl ether
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Carbonic Anhydrase
  • Recptor
    Carbonic Anhydrase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    6035-49-0
  • Formula Weight
    236.22
  • Molecular Formula
    C12H12O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL?(529.17 mM)
  • SMILES
    COc1cc2ccc(=O)oc2c(OC)c1OC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Davis R A Vullo D Maresca A et al. Natural product coumarins that inhibit human carbonic anhydrases[J]. Bioorganic & medicinal chemistry 2012 21(6):1539-1543.
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