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SR1001

CAS No. 1335106-03-0

SR1001( —— )

Catalog No. M19942 CAS No. 1335106-03-0

SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	81	In Stock
5MG	73	In Stock
10MG	140	In Stock
25MG	275	In Stock
50MG	491	In Stock
100MG	703	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

SR1001
Note

Research use only, not for human use.
Brief Description

SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).
Description

SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Nuclear Receptor/Transcription Factor
Target

ROR
Recptor

RORα| RORγ
Research Area

Neurological Disease
Indication

Multiple sclerosis

Chemical Information

CAS Number

1335106-03-0
Formula Weight

477.4
Molecular Formula

C15H13F6N3O4S2
Purity

>98% (HPLC)
Solubility

DMSO: 45 mg/mL;Ethanol: 45 mg/mL;Water: Insoluble
SMILES

CC(=O)Nc1nc(C)c(s1)S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Solt LA et al. Suppression of TH17 differentiation and autoimmunity by a synthetic ROR ligand. Nature. 2011 Apr 28;472(7344):491-4.

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