Cart
sales@molnova.com
Isoetharine mesylate salt
CAS No. 7279-75-6
Isoetharine mesylate salt( Isoetarine mesilate )
Catalog No. M19891 CAS No. 7279-75-6
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 28 | In Stock |
|
| 25MG | 46 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameIsoetharine mesylate salt
-
NoteResearch use only, not for human use.
-
Brief DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
-
DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.(In Vitro):Isoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.(In Vivo):Isoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
-
In VitroIsoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.
-
In VivoIsoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
-
SynonymsIsoetarine mesilate
-
PathwayAngiogenesis
-
TargetAdrenergic Receptor
-
Recptorβ-adrenergic receptor| PXR
-
Research AreaOthers
-
Indication——
Chemical Information
-
CAS Number7279-75-6
-
Formula Weight335.42
-
Molecular FormulaC14H25NO6S
-
Purity>98% (HPLC)
-
SolubilityDMSO:199.7 mM;Water:199.7 mM
-
SMILESCS(O)(=O)=O.CCC(NC(C)C)C(O)c1ccc(O)c(O)c1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Ratajewski M et al. Screening of a chemical library reveals novel PXR-activating pharmacologic compounds. Toxicol Lett. 2015 Jan 5;232(1):193-202.
molnova catalog
related products
-
ICI 89406
ICI 89406 is a β-adrenergic antagonist.
-
L-Adrenaline
L-Epinephrine(L-Adrenaline) is a hormone and a neurotransmitter.
-
Ajmalicine
Ajmalicine (Raubasine) is a potent adrenolytic agent which preferentially blocks α1-adrenoceptor. Ajmalicine is an reversible but non-competitive nicotine receptor full inhibitor, IC50 = 72.3 μM. Ajmalicine also can be used as anti-hypertensive, and serpentine, with sedative activity。
