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Talinolol
CAS No. 57460-41-0
Talinolol( (±)-Talinolol )
Catalog No. M27440 CAS No. 57460-41-0
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 48 | In Stock |
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| 2MG | 29 | In Stock |
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| 5MG | 44 | In Stock |
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| 10MG | 84 | In Stock |
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| 25MG | 188 | In Stock |
|
| 50MG | 323 | In Stock |
|
| 100MG | 553 | In Stock |
|
| 200MG | 802 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTalinolol
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NoteResearch use only, not for human use.
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Brief Description(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
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Description(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
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In VitroHuman OATP1A2-, rat Oatp1a5-, and rat Mdr1a-mediated Talinolol transport can be inhibited by naringin, with IC50s of 343, 12.7, and 604 μM, respectively, in LLC-PK1 cell and Xenopus laevis oocyte systems.
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In VivoTalinolol (20 mg/kg; i.p.) plasma and liver AUC0-5 h are increased by Zosuquidar administration.Bioavailability of Talinolol can be enhanced by coadministration with grapefruit juice (GFJ) in rats.
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Synonyms(±)-Talinolol
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number57460-41-0
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Formula Weight363.502
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Molecular FormulaC20H33N3O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (275.11 mM)
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SMILESCC(C)(C)NCC(O)COc1ccc(NC(=O)NC2CCCCC2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Asano T, Murayama T, Hirai Y, Shoji J. Comparative studies on the constituents of ophiopogonis tuber and its congeners. VIII. Studies on the glycosides of the subterranean part of Ophiopogon japonicus Ker-Gawler cv. Nanus. Chem Pharm Bull (Tokyo). 1993;41
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