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N-Methylcytisine
CAS No. 486-86-2
N-Methylcytisine( Caulophylline )
Catalog No. M18630 CAS No. 486-86-2
N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 50 | In Stock |
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| 2MG | 29 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 73 | In Stock |
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| 25MG | 140 | In Stock |
|
| 50MG | 222 | In Stock |
|
| 100MG | 330 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameN-Methylcytisine
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NoteResearch use only, not for human use.
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Brief DescriptionN-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).
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DescriptionN-Methylcytisine's nicotinic receptors have high affinity (KD = 5 nM)to nAChR from squid optical ganglia. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).
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In Vitro——
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In Vivo——
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SynonymsCaulophylline
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PathwayJAK/STAT Signaling
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TargetSTAT
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RecptorOthers
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Research AreaOthers-Field
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Indication——
Chemical Information
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CAS Number486-86-2
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Formula Weight204.27
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Molecular FormulaC12H16N2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 120 mg/mL (587.46 mM)
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SMILESCN1CC2CC(C1)C3=CC=CC(=O)N3C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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