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RO5454291
CAS No. ——
RO5454291( RO 5454291 )
Catalog No. M16939 CAS No. ——
RO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameRO5454291
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NoteResearch use only, not for human use.
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Brief DescriptionRO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.
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DescriptionRO5258638 is a small molecule inhibitor of CDK5-p25 protein-protein interaction with IC50 of 1.39 uM.
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In Vitro——
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In Vivo——
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SynonymsRO 5454291
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight357.458
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Molecular FormulaC19H27N5O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCCC(C)(C)C(N(C1)CC2=C1C(NC3=NC(OC)=CC=C3)=NN2)=O
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Chemical Name1-(3-((6-methoxypyridin-2-yl)amino)-6,6-dimethyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5(1H)-yl)-2,2-dimethylbutan-1-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bellón-Echeverría I, et al. Sci Rep. 2018 Mar 23;8(1):5083.
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