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Ketanserin tartrate
CAS No. 83846-83-7
Ketanserin tartrate( R41468 tartrate )
Catalog No. M16108 CAS No. 83846-83-7
A high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameKetanserin tartrate
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NoteResearch use only, not for human use.
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Brief DescriptionA high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
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DescriptionA high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C; also has a high affinity antagonist for the H1 receptor (Ki= 2 nM) and α1-adrenergic receptor (Ki=40 nM); an antihypertensive agent.Hypertension Approved.
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In Vitro——
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In Vivo——
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SynonymsR41468 tartrate
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PathwayGPCR/G Protein
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaCardiovascular Disease
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IndicationHypertension
Chemical Information
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CAS Number83846-83-7
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Formula Weight545.5136
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Molecular FormulaC26H28FN3O9
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Purity>98% (HPLC)
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SolubilityH2O: 30 mg/mL (Need ultrasonic and warming)
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SMILESO=C(N1CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)NC4=C(C=CC=C4)C1=O.O[C@H]([C@H](C(O)=O)O)C(O)=O
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Chemical Name2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-, (2R,3R)-2,3-dihydroxybutanedioate (1:1)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Creed-Carson M, et al. Behav Brain Res. 2011 Jun 1;219(2):273-9.
2. Catafau AM, et al. J Cereb Blood Flow Metab. 2010 May;30(5):985-93.
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