Enoxolone

CAS No. 471-53-4

Enoxolone( Arthrodont | Biosone | Enoxolone | α-Glycyrrhetinic Acid? | GM 1658 | NSC 35347 | PO 12 | STX 352 )

Catalog No. M14567 CAS No. 471-53-4

Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 28 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G 27 In Stock

Biological Information

  • Product Name
    Enoxolone
  • Note
    Research use only, not for human use.
  • Brief Description
    Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption.
  • Description
    Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the drug is used in various countries.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Arthrodont | Biosone | Enoxolone | α-Glycyrrhetinic Acid? | GM 1658 | NSC 35347 | PO 12 | STX 352
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Dehydrogenase
  • Recptor
    DHO
  • Research Area
    Other Indications
  • Indication
    ——

Chemical Information

  • CAS Number
    471-53-4
  • Formula Weight
    470.68
  • Molecular Formula
    C30H46O4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 94 mg/mL (199.71 mM)
  • SMILES
    CC(C)([C@](CC[C@@]([C@@]1(CC[C@]2(CC[C@](C(O)=O)(C[C@]2(C1=C3)[H])C)C)C)4C)5[H])[C@@H](O)CC[C@]5(C)[C@@]4([H])C3=O
  • Chemical Name
    (2S,4aS,6aS,6bR,8aR,10S,12aS,12bR,14bR)-10-hydroxy-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-2-carboxylic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Boldt J, et al. Expert Opin PharmacOthers. 2007, 8(13):2135-47.
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