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CFTR(inh)-172
CAS No. 307510-92-5
CFTR(inh)-172( CFTR(inh)-172 | Cystic Fibrosis Transmembrane Conductance Regulator Inhibitor 172 )
Catalog No. M13982 CAS No. 307510-92-5
CFTRinh-172 is a voltage-independent, selective CFTR inhibitor with Ki of 300 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 60 | In Stock |
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| 2MG | 36 | In Stock |
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| 5MG | 58 | In Stock |
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| 10MG | 93 | In Stock |
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| 25MG | 188 | In Stock |
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| 50MG | 352 | In Stock |
|
| 100MG | 519 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCFTR(inh)-172
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NoteResearch use only, not for human use.
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Brief DescriptionCFTRinh-172 is a voltage-independent, selective CFTR inhibitor with Ki of 300 nM.
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DescriptionCFTRinh-172 is a voltage-independent, selective CFTR inhibitor with Ki of 300 nM, showing no effects on MDR1, ATP-sensitive K+ channels, or a series of other transporters.
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In Vitro——
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In Vivo——
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SynonymsCFTR(inh)-172 | Cystic Fibrosis Transmembrane Conductance Regulator Inhibitor 172
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PathwayApoptosis
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TargetCFTR
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RecptorCFTR
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number307510-92-5
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Formula Weight409.4
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Molecular FormulaC18H10F3NO3S2
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Purity>98% (HPLC)
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SolubilityDMSO: 82 mg/mL (200.29 mM)
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SMILESO=C(O)C1=CC=C(/C=C(SC(N2C3=CC=CC(C(F)(F)F)=C3)=S)/C2=O)C=C1
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Chemical Name4-{[(5Z)-4-Oxo-2-sulfanylidene-3-[3-(trifluoromethyl)phenyl]-1,3-thiazolidin-5-ylidene]methyl}benzoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ma T, et al. J Clin Invest. 2002, 110(11), 1651-1658.
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