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Conivaptan

CAS No. 210101-16-9

Conivaptan( YM-087 | ZINC 12503187 )

Catalog No. M13330 CAS No. 210101-16-9

A potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively; has less potency for OT receptors and no effect on V1B receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Conivaptan
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively; has less potency for OT receptors and no effect on V1B receptor.
  • Description
    A potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively; has less potency for OT receptors and no effect on V1B receptor; blocks AVP-induced cAMP production of cultured renal epithelium cells concentration dependently and has no agonistic activities.Other IndicationApproved.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    YM-087 | ZINC 12503187
  • Pathway
    GPCR/G Protein
  • Target
    Vasopressin Receptor
  • Recptor
    Vasopressin Receptor
  • Research Area
    Other Indications
  • Indication
    Other Disease

Chemical Information

  • CAS Number
    210101-16-9
  • Formula Weight
    498.583
  • Molecular Formula
    C32H26N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC1=NC2=C(N1)CCN(C3=CC=CC=C32)C(=O)C4=CC=C(C=C4)NC(=O)C5=CC=CC=C5C6=CC=CC=C6
  • Chemical Name
    N-[4-[(4,5-Dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1,1'-Biphenyl]-2-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Tahara A, et al. J Pharmacol Exp Ther. 1997 Jul;282(1):301-8. 2. Tahara A, et al. Cardiovasc Res. 1998 Apr;38(1):198-205. 3. Nakayama S, et al. Neurocrit Care. 2016 Apr;24(2):273-82.
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