Lomitapide Mesylate

CAS No. 202914-84-9

Lomitapide Mesylate( —— )

Catalog No. M13157 CAS No. 202914-84-9

Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 84 In Stock
5MG 56 In Stock
10MG 92 In Stock
25MG 140 In Stock
50MG 221 In Stock
100MG 333 In Stock
200MG 491 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Lomitapide Mesylate
  • Note
    Research use only, not for human use.
  • Brief Description
    Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.
  • Description
    Lomitapide Mesylate is a potent microsomal triglyceride transfer protein (MTP) inhibitor, used in the treatment of familial hypercholesterolemia.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    CETP
  • Recptor
    MTP
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    202914-84-9
  • Formula Weight
    789.83
  • Molecular Formula
    C40H41F6N3O5S
  • Purity
    >98% (HPLC)
  • Solubility
    Ethanol: 100 mg/mL (126.6 mM); DMSO: 100 mg/mL (126.6 mM)
  • SMILES
    CS(O)(=O)=O.FC(F)(F)CNC(=O)C1(CCCCN2CCC(CC2)NC(=O)C2=CC=CC=C2C2=CC=C(C=C2)C(F)(F)F)C2=CC=CC=C2C2=CC=CC=C12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Davis KA, Miyares MA. Am J Health Syst Pharm. 2014 Jun 15;71(12):1001-8.
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