BRD-IN-17( —— )

Catalog No. M12999 CAS No. 1914047-59-8

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Get Quotation Bulk Inquiry Add to Cart

Product Name

BRD-IN-17
Note

Research use only, not for human use.
Brief Description

BRD-IN-17 is a cell permeable, family VIII bromodomain tool compound with additional PB1(2) activity over and above that of PFI-3.
Description

BRD-IN-17 is a cell permeable, family VIII bromodomain tool compound with additional PB1(2) activity over and above that of PFI-3; attenuates adipocyte differentiation and dramatically decreases lipid accumulation; a first in class chemical probe for Family VIII bromodomains.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Chromatin/Epigenetic
Target

Bromodomain
Recptor

Bromodomain
Research Area

——
Indication

——

CAS Number

1914047-59-8
Formula Weight

362.433
Molecular Formula

C21H22N4O2
Purity

>98% (HPLC)
Solubility

——
SMILES

——
Chemical Name

(E)-3-((6S,9R)-4-(cyclopropylamino)-6,7,8,9-tetrahydro-5H-6,9-epiminocyclohepta[d]pyrimidin-10-yl)-1-(2-hydroxyphenyl)prop-2-en-1-one

1. Gerstenberger BS, et al. J Med Chem. 2016 May 26;59(10):4800-11.

Calculator

molnova catalog