Bremelanotide

CAS No. 189691-06-3

Bremelanotide( PT-141 | PT 141 )

Catalog No. M12979 CAS No. 189691-06-3

A peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Bremelanotide
  • Note
    Research use only, not for human use.
  • Brief Description
    A peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction.
  • Description
    A peptide, non-selective melanocortin receptor agonist for treatment for female sexual dysfunction; selectively stimulates solicitational behaviors in the female rat, without affecting lordosis, pacing, or other sexual behaviors, does not cause generalized motor activation; a peptide analogue of α-MSH.Sexual Dysfunction Phase 3 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PT-141 | PT 141
  • Pathway
    GPCR/G Protein
  • Target
    Melanocortin Receptor
  • Recptor
    Melanocortin Receptor
  • Research Area
    Endocrinology
  • Indication
    Sexual Dysfunction

Chemical Information

  • CAS Number
    189691-06-3
  • Formula Weight
    1025.2
  • Molecular Formula
    C50H68N14O10
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCCCC(C(=O)NC1CC(=O)NCCCCC(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC1=O)CC2=CN=CN2)CC3=CC=CC=C3)CCCN=C(N)N)CC4=CNC5=CC=CC=C54)C(=O)O)NC(=O)C
  • Chemical Name
    N-Acetyl-L-norleucyl-L-alpha-aspartyl-L-histidyl-D-phenylalanyl-L-arginyl-L-tryptophyl-L-lysine (2-7)-lactam

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pfaus JG, et al. Proc Natl Acad Sci U S A. 2004 Jul 6;101(27):10201-4. 2. Molinoff PB, et al. Ann N Y Acad Sci. 2003 Jun;994:96-102. 3. Aughton KL, et al.
molnova catalog
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