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AM-630
CAS No. 164178-33-0
AM-630( AM 630 | AM630 | 6-Iodopravodoline )
Catalog No. M12488 CAS No. 164178-33-0
A potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 101 | In Stock |
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| 2MG | 44 | In Stock |
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| 5MG | 64 | In Stock |
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| 10MG | 92 | In Stock |
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| 25MG | 210 | In Stock |
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| 50MG | 338 | In Stock |
|
| 100MG | 538 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAM-630
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.
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DescriptionA potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1; inhibits forskolin-stimulated cyclic AMP production in CB1-transfected cells (22.6% at 1 uM and 45.9% at 10 uM).
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In Vitro——
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In Vivo——
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SynonymsAM 630 | AM630 | 6-Iodopravodoline
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number164178-33-0
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Formula Weight504.4
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Molecular FormulaC23H25IN2O3
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(C1=C(C)N(CCN2CCOCC2)C3=C1C=CC(I)=C3)C4=CC=C(OC)C=C4
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Chemical Name[6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ross RA, et al. Br J Pharmacol. 1999 Feb;126(3):665-72.
2. Malan TP Jr, et al. Pain. 2001 Sep;93(3):239-45.
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