K-Ras G12C-IN-1

CAS No. 1629265-17-3

K-Ras G12C-IN-1( —— )

Catalog No. M12441 CAS No. 1629265-17-3

A novel and irreversible inhibitor of mutant K-ras G12C.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 314 Get Quote
50MG 1791 Get Quote
100MG 3222 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
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Biological Information

  • Product Name
    K-Ras G12C-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    A novel and irreversible inhibitor of mutant K-ras G12C.
  • Description
    A novel and irreversible inhibitor of mutant K-ras G12C.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    Ras
  • Recptor
    Ras
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1629265-17-3
  • Formula Weight
    448.3423
  • Molecular Formula
    C22H23Cl2N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 40 mg/mL
  • SMILES
    COC1=C(C=C(C(=C1)Cl)C2=CC=CC=C2Cl)NCC(=O)N3CCN(CC3)C(=O)C=C
  • Chemical Name
    2-Propen-1-one, 1-[4-[2-[(2',6-dichloro-4-methoxy[1,1'-biphenyl]-3-yl)amino]acetyl]-1-piperazinyl]-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. From PCT Int. Appl. (2014), WO 2014152588 A1 20140925.
molnova catalog
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