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Bremelanotide acetate
CAS No. 1607799-13-2
Bremelanotide acetate( PT-141 acetate )
Catalog No. M12310 CAS No. 1607799-13-2
Bremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 62 | In Stock |
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| 10MG | 44 | In Stock |
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| 25MG | 79 | In Stock |
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| 50MG | 129 | In Stock |
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| 100MG | 193 | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBremelanotide acetate
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NoteResearch use only, not for human use.
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Brief DescriptionBremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.
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DescriptionBremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.Sexual Dysfunction Phase 3 Clinical(In Vivo):Bremelanotide Acetate (50-200 μg/kg; s.c.; once) significantly increases proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers.
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In Vitro——
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In VivoBremelanotide Acetate (50-200 μg/kg; s.c.; once) significantly increases proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers. Animal Model:Ovariectomized Long–Evans rats Dosage:50, 100, 200 μg/kg Administration:s.c.; once Result:Significantly increased proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers.
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SynonymsPT-141 acetate
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PathwayGPCR/G Protein
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TargetMelanocortin Receptor
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RecptorMelanocortin Receptor
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Research AreaEndocrinology
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IndicationSexual Dysfunction
Chemical Information
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CAS Number1607799-13-2
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Formula Weight1085.215
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Molecular FormulaC52H72N14O12
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 36 mg/mL
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SMILESCCCCC(C(=O)NC1CC(=O)NCCCCC(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC1=O)CC2=CN=CN2)CC3=CC=CC=C3)CCCN=C(N)N)CC4=CNC5=CC=CC=C54)C(=O)O)NC(=O)C.CC(=O)O
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Chemical Name(3S,6S,9R,12S,15S,23S)-12-((1H-imidazol-5-yl)methyl)-3-((1H-indol-3-yl)methyl)-15-((S)-2-acetamidohexanamido)-9-benzyl-6-(3-guanidinopropyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexaazacyclotricosane-23-carboxylic acid with acetic acid (1:1)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pfaus J, et al. J Sex Med. 2007 Nov;4 Suppl 4:269-79.
2. White WB, et al. J Hypertens. 2017 Apr;35(4):761-768.
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