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GW 841819X
CAS No. 146135-18-4
GW 841819X( GW841819X )
Catalog No. M11985 CAS No. 146135-18-4
GW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameGW 841819X
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NoteResearch use only, not for human use.
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Brief DescriptionGW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain.
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DescriptionGW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain that displays activity in vivo against NUT-midline carcinoma, multiple myeloma, mixed-lineage leukemia, and acute myeloid leukemia.
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In Vitro——
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In Vivo——
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SynonymsGW841819X
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research Area——
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Indication——
Chemical Information
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CAS Number146135-18-4
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Formula Weight487.94
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Molecular FormulaC26H22ClN5O3
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(OCC1=CC=CC=C1)N[C@H]2C3=NN=C(C)N3C4=CC=C(OC)C=C4C(C5=CC=C(Cl)C=C5)=N2
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Chemical Name(R)-benzyl (6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)carbamate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chung CW, et al. J Med Chem. 2011 Jun 9;54(11):3827-38.
2. Baud MG, et al. Science. 2014 Oct 31;346(6209):638-41.
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