PU-H54

CAS No. 1454619-13-6

PU-H54( PU H 54 )

Catalog No. M11959 CAS No. 1454619-13-6

A potent, selective Grp94 inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 110 Get Quote
10MG 177 Get Quote
25MG 410 Get Quote
50MG 605 Get Quote
100MG 860 Get Quote
500MG 1728 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PU-H54
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective Grp94 inhibitor.
  • Description
    A potent, selective Grp94 inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PU H 54
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    HSP
  • Recptor
    HSP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1454619-13-6
  • Formula Weight
    337.45
  • Molecular Formula
    C18H19N5S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (296.35 mM)
  • SMILES
    CC1=CC(C)=C(SC2=NC3=C(N)N=CN(CCCC#C)C3=N2)C=C1
  • Chemical Name
    8-((2,4-dimethylphenyl)thio)-3-(pent-4-yn-1-yl)-3H-purin-6-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Khandelwal A, et al. ACS Med Chem Lett. 2017 Sep 1;8(10):1013-1018. 2. Crowley VM, et al. J Med Chem. 2016 Apr 14;59(7):3471-88.
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